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Cetilistat (Oblean) i powder video
I-Cetilistat (i-Oblean) i-powder base-Characters
igama: | Cetilistat (Oblean) powder |
CAS: | 282526-98-1 |
Ifomula yeMolekyuli: | C25H39NO3 |
Ubunzima Ezinto: | 316.31 |
Melt Point: | 190-200 ° C |
Isitoreji sokugcina: | Ukushisa kwamagumbi |
umbala: | Grey Powder |
Yintoni i-Cetilistat powder?
I-Cetilistat, eyaziwa ngokuba yi-ATL-962, i-Oblean, okanye i-Citilistat, iyeza elitsha nelisebenzayo elenzelwe ukunyangwa kokukhuluphala. I-alkylamine derivative kunye ne-gastrointestinal lipase inhibitor ejolise ngokukodwa kwaye inqanda i-enzymes ejongene nokuphula amafutha okutya. Ngokuthintela ezi enzymes, i-cetilistat, enokuthi ithathwe kubaboneleli abathembekileyo abafana AASraw, kunciphisa ukunyuswa kwamafutha ekudleni, okukhokelela ekulahlekeni kwesisindo.
I-Cetilistat isetyenziswe ngokubambisana nekhalori ephantsi, i-fat-fat-fat diet kunye ne-regimen efanelekileyo yokuzivocavoca ukuququzelela ukulahleka kwesisindo. Eli chiza lichasene nokutyeba lithengiswa phantsi kwamagama eebhrendi ezahlukeneyo, kuquka iCetislim, iKilfat, i-Oblean, kunye neCheckwt.
Njengekhompawundi ye-benzoxazine, eyona ndlela iphambili yokwenza i-cetilistat ibandakanya ukuthintela ukugaywa kunye nokufunxwa kwamafutha okutya kwindlela ye-gastrointestinal, ekugqibeleni inceda abantu kuhambo lwabo lokuncipha. Nge-AASraw njengomthengisi othembekileyo, abantu abafuna izisombululo ezisebenzayo zokulahlekelwa kwesisindo banokufaka ngokuzithemba i-cetilistat kwirejimeni yabo.
Imbali emfutshane yeCetilistat (Oblean) powder
Imbali yophuhliso kunye nokuvunywa kwe-cetilistat ibuyele kwi-2013 xa iyeza lifumana imvume yalo yokuqala yokulawula ukutyeba eJapan. Ukutyhubela iminyaka, i-cetilistat iye yafumana ukuthandwa kumazwe ahlukeneyo kwihlabathi liphela ngenxa yokusebenza kwayo kunye nokunyamezelana ekunyangeni ukutyeba.
Ukusetyenziswa kwePowder yeCetilistat(Oblean) kwaye isebenza njani?
(1)Ukujolisa kwi-lipases yesisu
I-Cetilistat isebenza ngokujolisa kwi-lipases ye-gastrointestinal, eyi-enzymes ejongene nokuphula kunye nokugaya amafutha emzimbeni womntu.
(2)Ukuthintela ukucolwa kwamafutha kunye nokufunxa
Ngokuthintela ezi lipases, i-cetilistat ikhusela ukuphuka kunye nokufunxa kwamafutha kwindlela yesisu. Amafutha angagaywanga akhutshwa emzimbeni ngelindle. Le nkqubo ikhokelela ekunciphiseni kwekhalori yokutya kwaye ekugqibeleni ibangele ukulahleka kwesisindo.
Ziziphi iiNzuzo zeCetilistat (Oblean) powder?
I-Cetilistat(Oblean) inikezela ngothotho lweenzuzo kubantu abafuna ulawulo olusebenzayo lokutyeba. Njengechiza elinamandla lokunciphisa umzimba kunye ne-anti-obesity agent, ayincedi kuphela ekunciphiseni ubunzima kodwa ibonelela ngeenzuzo ezininzi ezongezelelweyo eziyahlula kwamanye amayeza okunciphisa umzimba. Ezinye zeenzuzo eziphambili ze-cetilistat ziquka:
(1) Ukuxhasa impilo enempilo ngokuncipha
I-Cetilistat iyanciphisa ngokukhawuleza ukuqokelela kwamafutha emzimbeni, inceda ukugcina i-BMI enempilo kunye nokunciphisa amathuba okuba neemeko ezisongela ubomi ezinxulumene nokukhuluphala, njengohlobo lwe-2 yeswekile, isifo senhliziyo, uxinzelelo lwegazi oluphezulu, kunye nomhlaza othile.
(2) Ukuphucula ukwehla kobunzima kunye nokunciphisa i-hemoglobin ye-glycosylated kwisigulana seswekile esityebileyo
Izifundo zeklinikhi zibonise ukusebenza kwe-cetilistat ekunciphiseni ubunzima kunye namanqanaba e-glycosylated hemoglobin (HbA1c) kwizigulane ezityebileyo ezinesifo sikashukela sohlobo lwe-2, ukubonelela ngolawulo olungcono lweswekile.
(3)Ukunyamezela kunye nokhuseleko
I-Cetilistat ngokuqhelekileyo inyamezeleke kakuhle, kunye nemiphumo engathandekiyo ukuya kwimodareyitha ehlala iyancipha ngokusetyenziswa okuqhubekayo. Xa kuthelekiswa namanye amachiza okunciphisa umzimba, njenge-orlistat, i-cetilistat ifunyenwe ukuba ibangele imiphumo embalwa kwaye ingaphantsi.
(4) Ukufezekiswa okukhawulezileyo kweenjongo zokunciphisa umzimba
Ngelixa amanye amayeza achasene nokutyeba kakhulu afuna ixesha elide ukuze afezekise ukwehla kobunzima obukhulu, i-cetilistat inokunikezela ngeziphumo ezinqwenelekayo phakathi kweeveki ezimalunga ne-12 xa isetyenziswa kunye nokutya okunamafutha aphantsi kunye nerejimeni yokuzilolonga rhoqo.
(5) Ukunciphisa i-cholesterol enokwenzeka
I-Cetilistat inokunceda ukunciphisa i-cholesterol epheleleyo kunye namanqanaba e-cholesterol ye-LDL, ngaloo ndlela igalelo ekuphuculeni impilo ye-cardiovascular and ukunciphisa ingozi yesifo senhliziyo.
(6) Ukunciphisa umngcipheko wesifo senhliziyo
Ngokujongana nokutyeba kakhulu kunye nokukhuthaza ukutya okunempilo, i-cetilistat inokunciphisa umngcipheko wesifo senhliziyo. Uphononongo lweeveki ze-12 olungenamkhethe, oluyimfama olubandakanya izigulane ezityebileyo ezine-diabetes mellitus lubonise ukunciphisa ubunzima, ukuphuculwa kokulawulwa kwe-glycemic, kunye nokunciphisa umjikelezo wesinqe, umngcipheko wesifo senhliziyo.
(7)Ukwehlisa uxinzelelo lwegazi
Njengoko i-cetilistat iququzelela ukulahleka kwesisindo, inokukhokelela ekunciphiseni uxinzelelo lwegazi, inceda ukukhusela uxinzelelo lwegazi kunye nemingcipheko yempilo ehambelana nayo njenge-stroke, isifo sezintso, kunye nesifo sesibindi.
Xa ifunyenwe kubathengisi abathembekileyo njenge-AASraw, i-cetilistat isebenza njengesixhobo esixabisekileyo ekukhuthazeni indlela yokuphila enempilo kunye nokujongana nemingeni yokukhuluphala. Ngokubandakanya i-cetilistat kwisicwangciso esibanzi sokulawula ubunzima, abantu ngabanye banokuyonwabela ezi zibonelelo kwaye basebenze ekuphuculeni impilo yonke.
Usetyenziso lwezonyango lweCetilistat(Oblean)
(1)Unyango lokutyeba kubantu abadala
I-Cetilistat isetyenziselwa ukunyanga ukukhuluphala kubantu abadala. Ngokuqhelekileyo imiselwe ecaleni kwekhalori encitshisiweyo, ukutya okunamafutha aphantsi kunye nerejimeni yokuzivocavoca rhoqo ukwandisa ukusebenza kwayo.
(2)Ulawulo lweengxaki ezinxulumene nokutyeba
Ukongeza ekukhuthazeni ukulahleka kwesisindo, i-cetilistat nayo ibonakaliswe ukuphucula i-comorbidities ehlobene nokukhuluphala, njengale:
①Uhlobo lwesi-2 seswekile
I-Cetilistat inokunceda ekuphuculeni ulawulo lwe-glycemic kwizigulane ezityebileyo ezinesifo sikashukela sohlobo lwe-2 ngokunciphisa ubunzima bomzimba kunye nokunciphisa amanqanaba e-glycosylated hemoglobin (HbA1c).
②I-cholesterol ephezulu
I-Cetilistat iboniswe ukunciphisa amanqanaba e-cholesterol epheleleyo kunye ne-low-density lipoprotein (LDL) ye-cholesterol, eyaziwa nangokuthi "i-cholesterol embi", enokufaka isandla ekuphuhliseni izifo zentliziyo.
③Uxinzelelo lwegazi
Ukunciphisa umzimba okuphunyezwe nge-cetilistat kunokunceda ukunciphisa uxinzelelo lwegazi kubantu abatyebileyo, ukunciphisa umngcipheko wokuphuhlisa uxinzelelo lwegazi kunye neengxaki ezinxulumene nazo.
Ikuphatha njani uCetilistat(Oblean) ukutyeba?
Ukutyeba kakhulu yenye yeengxaki zempilo yoluntu ezikhoyo namhlanje. Sisifo esintsonkothileyo, esinganyangekiyo kunye nesinokuphazamiseka kwimisebenzi emininzi ebonakaliswa kukuqokelelwa kwamafutha / izicubu zeadipose.
Ukutyeba kakhulu kunxulunyaniswa nokuphazamiseka kwempilo enje ngohlobo lweswekile 2, uxinzelelo lwegazi, ihyplipidemia, icholesterol ephezulu, umhlaza othile, kunye nesifo sentliziyo esifana nokubetha kunye nokuphazamiseka kwentliziyo.
Ukutyeba kumazwe amaninzi kuye kwafikelela kubhubhane kwaye ngenxa yoko inkxalabo yezempilo kwihlabathi liphela.
Uphando lubonisa ukuba ukulahlekelwa ubunzima obuzinzileyo ukusuka kwi-5 ukuya kwi-10% yobunzima bomzimba wakho bokuqala kunokunciphisa kakhulu ukuphazamiseka kwe-metabolic ezinxulumene nokutyeba. Ii-Anti-obesity agents zidla ngokunyusa inkcitho yamandla ngoko ke ukwehla kobunzima ngolawulo lwe-neural kunye ne-metabolic. I-Cetilistat yi-gastrointestinal pancreatic lipase inhibitor eyi-agent esebenzayo yokulwa nokutyeba kwizifundo zabantu.
I-Cetilistat isebenza ngokuthintela ukugaya kunye nokufunxa kwamafutha ngaphakathi kokutya okutyayo. Xa amanqatha engacolwanga akhutshelwa ilindle xa kuthuthwa amathumbu. Ifezekisa oku ngokuvimbela i-enzyme lipases ejongene nokuphula i-triglycerides (i-fat / lipid emzimbeni) emathunjini.Imiphumo ye-cetilistat ngoko ibonakaliswe kwindlela yesisu. Yiyo ke loo nto ithetha ukuba i-cetilistat yahlukile kwezinye iiarhente ezichasene nokutyeba eziphembelela ingqondo yakho ukunciphisa umdla wokutya kuba isebenza kwi-periphery.
Xa ukugaya kunye nokufunxa kwamafutha okutya kuthintelwe, ukuchithwa kwamafutha kunqunyelwe ngoko ke inkcitho ephantsi yamandla ibangela ukulahleka kwesisindo. Nangona, i-Cetilistat iya kukunceda ulahlekelwe isisindo phezu kwakho ukugcina ukutya okunesondlo okuncinci okuhamba kunye nokuzivocavoca umzimba. ulawulo lokutyeba ngempumelelo.
Ngaba i-Cetilistat (Oblean) ipowder inayo nayiphi na i-Side Effects?
Izigulane ezifumana unyango lokukhuluphala kunye ne-Cetilistat powder zingabandezeleka kwimiphumo emibi. Kufuneka uxelele ugqirha wakho ukuba oku kuyenzeka. Eminye imizekelo inikwe apha:
▪Ukutyeba elindle
▪Intlungu yesisu
▪Iflatus ephumayo
▪Ukubona amafutha
▪Ukungakwazi ukuzibamba kwamathumbu
▪Ukuqunjelwa
▪Iingqaqambo Zesisu
▪Urhudo
▪Izitulo ezithambileyo
▪Ukuxinana kweempumlo
▪Ukuzithuma rhoqo
▪Intlungu esiswini
Nangona ukuphendula okunomdla ngokuqhelekileyo kuthathwa njengento eqhelekileyo, iziganeko ezimbi kakhulu zingenzeka. Buza udokotela wakho ngokukhawuleza ukuba oko kwenzeka.
Cetilistat vs Orlistat
(1)Ukufana kwindlela yokwenza
I-Cetilistat kunye ne-Orlistat yabelana ngendlela efanayo yokusebenza, zombini ijolise kwaye inqanda i-lipases yamathumbu ukunciphisa ukuxutywa kwamafutha kunye nokukhuthaza ukulahleka kwesisindo.
(2)Umahluko kwisakhiwo sekhemikhali kunye neempawu
Nangona iindlela zabo zesenzo zifana, i-cetilistat kunye ne-Orlistat ziyahluka kwizakhiwo zabo zeekhemikhali, ezikhokelela ekuhlukeni kwiimpawu zabo ze-pharmacokinetic kunye neeprofayili zempembelelo.
(3) Ukuthelekisa ukusebenza kunye neziphumo zokulahleka kwesisindo
Izilingo zeklinikhi ziye zabonisa ukuba i-cetilistat ifaniswa ne-Orlistat ngokubhekiselele ekusebenzeni kokulahlekelwa kwesisindo. Omabini amayeza anokunceda izigulana zifezekise ukuncipha okukhulu kobunzima xa zisetyenziswa njengenxalenye yenkqubo yokulawula ukutyeba.
(4) Ukunyamezela kunye nothelekiso lweprofayili yecala
I-Cetilistat ngokubanzi ineprofayili yokunyamezela ngakumbi xa kuthelekiswa ne-Orlistat. Izigulane ezithatha i-cetilistat azinakwenzeka ukuba zibe nemiphumo emibi yesisu, okwenza kube yinto ekhangayo ngakumbi kwabo banobunzima bokunyamezela i-Orlistat.
Indlela yokusebenzisa i-Cetilistat (oblean) powder ngokukhuselekileyo?
(1)Idosi ecetyiswayo kunye nezikhokelo zolawulo
I-Cetilistat ngokuqhelekileyo imiselwe kwi-dosage ye-60 mg, ithathwe kathathu ngosuku ngokutya. Kufuneka ithathwe ngokukhawuleza ngaphambi, ngexesha, okanye ukuya kuthi ga kwiyure enye emva kwesidlo ngasinye esiphambili. Ukuba ukutya kuphosakele okanye akunamafutha, idosi inokugqithwa.
(2)Ukunyangwa kunye nezilumkiso
Abantu abathile akufanele bathathe i-cetilistat, kubandakanywa nalabo abane-syndrome ye-malabsorption engapheliyo, i-cholestasis, okanye i-hypersensitivity kuyo nayiphi na into yamachiza. Abasetyhini abakhulelweyo okanye abancancisayo kufuneka badibane nomboneleli wabo wezempilo ngaphambi kokusebenzisa i-cetilistat. Izigulana ezineemeko zonyango ezikhoyo okanye abo bathatha amanye amayeza kufuneka baxoxe ngobungozi obunokubakho kunye neenzuzo kunye nomboneleli wabo wezempilo.
(3)Ukunxibelelana kweziyobisi okunokwenzeka
I-Cetilistat (oblean) inokusebenzisana namayeza athile, kuquka i-anticoagulants, amayeza esifo seswekile, kunye neyeza ze-thyroid. Izigulana kufuneka zazise umboneleli wabo wezempilo malunga nawo onke amayeza kunye nezongezelelo abazenzayo ngoku ukuphepha ukusebenzisana okunokwenzeka.
(4)Ukubeka iliso kunye nokulandelwa ngexesha lonyango
Ukubeka iliso rhoqo kunye nokuqeshwa okulandelwayo kunye nomboneleli wezempilo kubalulekile ngexesha lonyango lwe-cetilistat. Ezi ziqendu zivumela ukuhlolwa kwenkqubela yonyango, ulawulo lwempembelelo yecala, kunye nohlengahlengiso olunokubakho lwedosi ukuba kuyimfuneko.
Kuphi ukuthenga i-Cetilistat (Oblean) powder?
Kukho imithombo emininzi ye-Cetilistat powder ethengiswa kwi-intanethi kwiimarike, kwaye kukho imithombo emininzi ekhohlisa abathengi ngeemveliso zomgunyathi. Ukuba ufuna ukuthenga ubuninzi be-Cetilistat (oblean) ipowder okanye i-powder ephezulu ye-Cetilistat ethengiswayo, i-Cetilistat enokwethenjelwa kwaye ehloniphekileyo umenzi wepowder yeCetilistat / umthengisi / i-factory / umthengisi yinto efanelekileyo. Unokukhangela uphononongo oluhle okanye olubi malunga nabo kwi-intanethi, okuya kukunceda wenze ukhetho olufanelekileyo. Ukuba ukhangele umthengisi we-Cetilistat onokwethenjelwa kunye nothembekileyo, ngoko i-AASraw iyona nto ikhethekileyo.
Njengomkhiqizi omnye othembekileyo we-Cetilistat powder e-China, i-AASraw ivelisa zonke iikhompawundi ngokungqongqo ngokuhambelana nezikhokelo ze-cGMP kwaye isebenze iyunithi yokuvelisa i-FDA evunyiweyo ye-state-of-art ukuqinisekisa ukucoceka okuphezulu. I-AASraw inomzi wayo ozimeleyo we-Cetilistat powder, iziko lophando kunye nophuhliso. Inkqubo yabo yokubonelela nge-powder ye-Cetilistat izinzile kwaye iyakwazi ukufumana ii-odolo zokuthengisa kunye ne-wholesale ye-bulk Cetilistat powder. Ukongezelela, i-AASraw inokubonelela ngexabiso elikhuphisanayo le-Cetilistat powder kwimarike kulabo bafuna ukuthenga i-Cetilistat powder.
Xa uyala ukusuka kwi-AASraw, unokuqiniseka ukuba iphakheji nganye ye-Cetilistat powder, nokuba yeyokuthengisa okanye inqwaba ye-Cetilistat powder, iya kuthunyelwa ngaphandle kwexesha kwaye ihanjiswe ngokukhuselekileyo. Ukongezelela, i-AASraw inokuthumela i-Cetilistat powder kuyo yonke indawo kwihlabathi, kuquka i-USA, iCanada, iMexico, iYurophu kunye ne-Australia. Musa ukuthatha amathuba ngempilo yakho okanye imali yakho - khetha i-AASraw njengomthengisi wakho we-Cetilistat (oblean) wepowder kwaye ufumane uxolo lwengqondo oluza kunye nokusebenza kunye nomvelisi we-powder othembekileyo we-Cetilistat.
I-Cetilistat powder (282526-98-1) -COA
I-Cetilistat powder (282526-98-1) -COA
Indlela yokuthenga i-Oblean powder: Thenga i-Cetilistat powder esuka kwi-AASraw
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Umbhali weli nqaku:
UGqr Monique UHong uthweswe isidanga kwiKholeji yase-UK Imperial yaseLondon kwiFakhalthi yezoNyango
Umbhali wephepha leJenali yeNzululwazi:
1. uNahid Shahabadi
IZiko loPhando lweBiology yezoNyango, iZiko leTekhnoloji yezeMpilo, iYunivesithi yaseKermanshah yeSayensi yezoNyango, eKermanshah, e-Iran
2. UWilliam E. Acree Omnci
ISebe leKhemistry, iYunivesithi yaseNorth Texas, i-1155 Union Circle Drive #305070, Denton, TX 76203, USA
3. Shuofeng Yuan
Iziko leVirology, iVaccinology kunye neTherapeutics, [imeyile ikhuselwe], IYunivesithi yaseHong Kong, iNgingqi yoLawulo oluKhethekileyo lwaseHong Kong
4. Padwal R
Uluvo lwangoku kwiZiyobisi zoPhando (London, England : 2000)
5. Ingca J
YaseBrazil, eSpain
Lo gqirha/ingcali yenzululwazi ayinakuvuma okanye ithethelele ukuthengwa, ukuthengiswa, okanye ukusetyenziswa kwale mveliso nangasiphi na isizathu. I-Aasraw ayinayo indibaniselwano okanye ubudlelwane, ichazwa okanye ngenye indlela, kunye nalo gqirha. Injongo yokucaphula lo gqirha kukuvuma, ukuvuma kunye nokuncoma uphando olupheleleyo kunye nomsebenzi wophuhliso owenziwe ngoososayensi abasebenza kule nto.