Ingcaciso yeMveliso
Ividiyo yeTadalafil Powder-AASraw
Tadalafil Powder Basic Characters
igama: | Tadalafil (Cialis) powder |
CAS: | 171596-29-5 |
I-molecular Formula: | C22H19N3O4 |
Isisindo somzimba: | 389.4 |
Melt Point: | 298-300 ° C |
Isitoreji sokugcina: | 20ºC |
umbala: | Powder |
Yintoni iTadalafil Powder?
I-Tadalafil Powder liyeza elisetyenziselwa ukuphatha i-erectile dysfunction (ED) kunye ne-pulmonary arterial hypertension (PAH). I-phosphodiesterase type 5 (PDE5) inhibitor esebenza ngokukhulula izihlunu emithanjeni yegazi, evumela ukunyuka kwegazi kwiindawo ezithile zomzimba. I-Tadalafil yaqala ukuvunywa yi-FDA kwi-2003 phantsi kwegama le-brand Cialis kwaye sele ibe yinto ekhethiweyo yonyango kumadoda ane-ED. I-Tadalafil ikwafumaneka njengamayeza aqhelekileyo, okwenza ukuba ifikeleleke kwaye ifikeleleke kwabo bayidingayo. Ifomu yePowder yeTadalafil ingasetyenziselwa iinjongo zophando okanye ukudibanisa amayeza. Kubalulekile ukuthenga i-Tadalafil Powder ngesiqinisekiso somgangatho. I-Cialis ifumaneka phantse kuzo zonke iikhemesti zengingqi kunye ne-intanethi kodwa izigulane kufuneka zibe ne-prescription ukuze zikwazi ukuyithenga. I-Tadalafil Powder eluhlaza ayifuni i-prescription. Unokuthenga i-Tadalafil Powder eluhlaza kwi-AASRAW. Umthengisi we-AASRAW unikezela ngePowder ephezulu yeTadalafil ngexabiso elifanelekileyo.
Isebenza njani iTadalafil Powder?
I-Tadalafil Powder luhlobo lwe-phosphodiesterase uhlobo lwe-5 (PDE5) inhibitor. Kwimeko ye-erectile dysfunction (ED), i-Tadalafil Powder isebenza ngokunyusa ukuhamba kwegazi kwi-penis, enokunceda indoda ifezekise kwaye igcine i-erection ngexesha lomsebenzi wesondo. Esi siphumo sixutyushwa ngokukhululeka kwemisipha egudileyo kwimithambo yegazi yepenis, evumela ukunyuka kwegazi kwindawo.
Kwimeko ye-pulmonary arterial hypertension (PAH), i-Tadalafil Powder isebenza ngokunciphisa uxinzelelo lwegazi kwimibhobho enika imiphunga. Oku kufezekiswa ngokuphumla kwezihlunu ezigudileyo kwimithambo yegazi yemiphunga, evumela ukunyuka kwegazi kunye nokuphucula i-oxygen.
Kubalulekile ukuba uqaphele ukuba i-Tadalafil Powder ayisebenzi ngaphandle kokuvuselela ngokwesondo. Ukuvuselela ngokwesondo kuyimfuneko ukuqalisa ukukhululwa kwe-nitric oxide (NO), leyo ivuselela ukuveliswa kwe-cGMP. I-Tadalafil Powder ke isebenza ngokuthintela i-PDE5 kunye nokuvumela ukunyuka kwamanqanaba e-cGMP ukukhuthaza ukukhululeka kwemisipha egudileyo kwimithambo yegazi.
Ukusetyenziswa kwamachiza eTadalafil Powder
I-Tadalafil Powder ingasetyenziselwa ukwenza iipilisi zomlomo okanye iipilisi zokunyanga i-ED okanye i-PAH. Ikwasetyenziswa ngamanye amaxesha kwizifundo zophando.
· Unyango lwe-erectile dysfunction (ED)
I-ED yimeko eqhelekileyo apho indoda inobunzima bokuphumelela okanye ukugcina i-erection ngexesha lomsebenzi wesondo. I-Tadalafil Powder isebenza ngokuvimbela i-enzyme ye-PDE5, ejongene nokuphula i-cGMP, i-molecule ekhuthaza ukukhululeka kwemisipha epholileyo kwi-penis kunye nokwandisa ukuhamba kwegazi kwindawo. Ngokuthintela i-PDE5, i-Tadalafil Powder inokunyusa amanqanaba e-cGMP kunye nokuphucula umsebenzi we-erectile. I-Tadalafil Powder idla ngokumiselwa njengeyeza lemihla ngemihla kunyango lwe-ED.
· Unyango lwe-pulmonary arterial hypertension (PAH)
I-PAH yimeko enqabileyo apho uxinzelelo lwegazi kwimithambo ehambisa imiphunga luphezulu ngendlela engaqhelekanga. Oku kunokukhokelela ekuphefumleni, ukudinwa, kunye nezinye iimpawu. I-Tadalafil Powder ikwayi-PDE5 inhibitor, kwaye isebenza ngokuphumla izihlunu ezigudileyo kwimithambo yegazi yemiphunga, eyehlisa uxinzelelo lwegazi kule mithambo. Oku kuvumela intliziyo ukuba impompe igazi ngokufanelekileyo kwaye iphucule iimpawu ze-PAH. I-Tadalafil Powder idla ngokuphathwa njengeyeza kanye ngosuku unyango lwe-PAH.
Ngaphandle kokusetyenziswa kwayo okuphambili, i-Tadalafil Powder iphinde iphandwe kwezinye izicelo ezinokubakho zonyango, ezifana nokunyangwa kwe-benign prostatic hyperplasia (BPH) kunye neempawu ezisezantsi ze-urinary tract (LUTS) kumadoda. Nangona kunjalo, oku kusetyenziswa akukavunywa yi-FDA kwaye uphando oluninzi luyafuneka ukuze kuqondwe ngokupheleleyo ukusebenza kwabo kunye nokhuseleko.
I-Tadalafil Powder iindlela ezahlukeneyo zokulawula (iipilisi zomlomo, ii-capsules, ii-injection, njl.)
I-Tadalafil Powder ngokuqhelekileyo ifumaneka ngendlela ye-crystalline Powder emhlophe, ethi emva koko yenziwe kwiifom ezahlukeneyo zedosi yokulawula. Iindlela ezahlukeneyo zolawulo lweTadalafil Powder ziquka:
Iipilisi zomlomo: I-Tadalafil Powder inokuqulunqwa kwiipilisi zomlomo, ezinokuthi zithathwe kunye okanye ngaphandle kokutya. Iipilisi zifumaneka kwiidosi ezahlukeneyo, kubandakanywa i-2.5mg, 5mg, 10mg, kunye ne-20mg, kwaye zithathwa njengoko ziyimfuneko kunyango lwe-erectile dysfunction (ED), okanye njengeyeza lemihla ngemihla unyango lwe-pulmonary arterial hypertension (PAH). ).
Iipilisi: I-Tadalafil Powder inokuphinda iqulunqwe kwii-capsules, ezithathwa ngokuqhelekileyo ngomlomo kunye okanye ngaphandle kokutya. Iipilisi kunokuba lula ukuginya kuneepilisi kwezinye izigulane, kwaye zinokufumaneka kwiidosi ezahlukeneyo ngokuxhomekeke kusetyenziso olucetywayo.
Iipilisi ezingaphantsi kweelwimi: I-Tadalafil Powder inokuqulunqwa kwiipilisi ezingaphantsi kweelwimi, ezibekwe phantsi kolwimi kwaye zivunyelwe ukuba zichithe. Olu hlobo lweTadalafil lunokuqala ngokukhawuleza kwesenzo xa kuthelekiswa namacwecwe omlomo, njengoko iyeza lifakwe ngokuthe ngqo kwigazi ngokusebenzisa i-mucous membranes emlonyeni.
Ifilimu ye-Buccal: I-Tadalafil Powder nayo inokuqulunqwa kwifilimu ye-buccal, efakwe ngaphakathi kwesihlathi kwaye ivumeleke ukuba ichithe. Olu hlobo lwe-Tadalafil lunokuthi lube nokuqala ngokukhawuleza kwesenzo xa kuthelekiswa namacwecwe omlomo, njengoko iyeza lifakwe ngokuthe ngqo kwigazi ngokusebenzisa i-mucous membranes emlonyeni.
I-injection: I-Tadalafil Powder inokuqulunqwa kwifomu yokutofa unyango lwe-pulmonary arterial hypertension (PAH). Olu hlobo lweTadalafil lulawulwa yingcali yezempilo ngenaliti kwi-vein okanye phantsi kwesikhumba.
Kubalulekile ukuba uqaphele ukuba iindlela ezahlukeneyo zeTadalafil zinokuba ne-dosing eyahlukeneyo kunye nemiyalelo yokulawula, kwaye izigulane kufuneka zilandele imiyalelo enikezwa ngumboneleli wabo wezempilo. Ukongezelela, izigulane kufuneka zixelele umboneleli wabo wezempilo nangaliphi na iyeza okanye izongezo ezithathayo ngaphambi kokuba baqale unyango nge-Tadalafil Powder, njengoko amanye amayeza angasebenzisana ne-Tadalafil Powder kunye nokwandisa umngcipheko wemiphumo emibi.
Umthamo kunye nokulawulwa kweTadalafil Powder
I-dosage kunye nokulawulwa kwe-Tadalafil Powder kuya kuxhomekeka kwimeko ethile ephathwayo, kunye nezinto ezigulayo ngamnye ezifana nobudala, ubunzima, kunye nembali yonyango. Kubalulekile ukulandela i-dosage kunye nemiyalelo yokulawula enikezelwa ngumboneleli wezempilo nokuba uthenge i-Tadalafil Powder eluhlaza kumenzi othembekileyo, kwaye ungagqithisi idosi ecetyiswayo. Imilinganiselo ekhoyo ye-Cialis (i-Tadalafil Powder) iquka i-2.5, i-5, i-10, kunye ne-20 mg.
Kunyango lwe-erectile dysfunction (ED), i-dose yokuqala ye-Tadalafil Powder yi-10mg, ithathwe ngomlomo njengoko ifunekayo, ngaphambi komsebenzi wesondo. Ukwandisa ukusebenza kwe-Cialis, kamva kunokulungiswa ngokuhambelana nokuqina kokuphendula kunye nokunyamezela ngokunciphisa kwi-5 mg okanye ukuyiphakamisa kwi-20 mg. I-Tadalafil Powder inokuthatyathwa kunye okanye ngaphandle kokutya, kodwa kufuneka ithathwe malunga nexesha elifanayo ngosuku ngalunye ukugcina amanqanaba angaguqukiyo emzimbeni. Kubalulekile ukuba uqaphele ukuba ukuvuselela ngokwesondo kuyadingeka ukuze i-Tadalafil Powder isebenze.
Kunyango lwe-pulmonary arterial hypertension (PAH), idosi yokuqala ye-Tadalafil Powder yi-40mg kanye yonke imihla, ithathwe ngomlomo kunye okanye ngaphandle kokutya. Idosi inokulungiswa ngokusekelwe kwimpendulo yomntu kunye nokunyamezela, kwaye izigulane kufuneka zibekwe esweni ngokusondeleyo kwimiphumo emibi.
I-Tadalafil Powder kufuneka ithathwe njengoko iyalathwa ngumboneleli wezempilo, kwaye izigulane akufanele zithathe i-dose engaphezu kweyodwa kwixesha leeyure ze-24 nokuba uthenge i-Tadalafil Powder eluhlaza kunye nomenzi we-AASRAW, kuba ubunyulu bu> 99.9%. Kwimeko yokugqithisa, izigulane kufuneka zifune unyango ngokukhawuleza.
Kubalulekile ukuba uqaphele ukuba i-Tadalafil Powder inokusebenzisana namayeza athile, kuquka i-nitrate, i-alpha-blockers, kunye ne-antibiotics ethile kunye neyeza ezichasayo. Izigulane kufuneka zixelele umboneleli wabo wezempilo kuwo onke amayeza kunye nezongezelelo abazithathayo ngaphambi kokuba baqale unyango ngeTadalafil Powder.
Yiba Nolindelo Olusengqiqweni
Ayingawo onke amayeza asebenzayo kuye wonke umntu. I-Tadalafil Powder lichiza elisebenzayo ngokubanzi, kodwa oku akuthethi ukuba i-slam-dunk ikulungele ngokufanelekileyo. Ngokutsho koncwadi lwenzululwazi, ukuba isebenza ngokukhawuleza kwaye isebenza njani inokwahluka.
Ngokomzekelo, iyeza linokuba luncedo kwiiyure ezingama-24 ukuya kwezingama-36 emva kokulawulwa, kwaye ukuya kuthi ga kwiiyure ezingama-72. Ke inokusebenza kuwe usuku lonke, ngelixa inokusebenza kumfana olandelayo kangangeentsuku ezintathu.
Ngaphezu koko, uphando oluthile lufumene ukuba i-20mg ye-Tadalafil inezinga le-52 yepesenti yokusebenza emva kwemizuzu ye-30, ebonisa ukuba amanye amadoda awakwazi ukuba neentlobano zesini kunye nesiqingatha seyure emva kokuyithatha.
Into enye ekufuneka uyikhumbule malunga nokusebenza kweCialis: ayivelisi ukumiswa kwangoko kunye nendalo. Ngenxa yokuba i-PDE5 inhibitors ayichaphazeli ngokuthe ngqo imisipha egudileyo yepenis (kodwa kunoko ithembele ekukhululweni kokuqala kwe-NO), ukuvuselela ngokwesondo kusafuneka ngaphambi kokuba i-penis yakho iqine.
Ziziphi iziphumo zecala le-Tadalafil Powder?
Njengawo nawaphi na amayeza, kubalulekile ukuba uqaphele imiphumo enokubakho kunye nezilumkiso xa uthatha i-Tadalafil Powder okanye i-Cialis.
(1)Iimpembelelo zecala leTadalafil Powder:
Iziphumo eziqhelekileyo zecala le-Tadalafil Powder ziquka:
intloko ebuhlungu
Umqolo obuhlungu
Iintsimbi zomzimba
Ukuqhuma
Ukunyanzelisa
Impumlo okanye impumlo egudileyo
Iziphumo ebezingalindelekanga ezimbalwa zinokubandakanya:
Isiyezi okanye ukukhanya kwentloko
I-priapism, i-erection ebuhlungu ehlala ixesha elide kuneeyure ze-4, ezinokubangela umonakalo wezicubu
uxinzelelo lwegazi oluphantsi
utshintsho kwindlebe kunye nombono
Intlungu yesifuba okanye ukubetha kwentliziyo okungaqhelekanga
Ukuphefumula okufutshane okanye ukudumba ezandleni, emaqatheni, okanye ezinyaweni
Ukuba ufumana naziphi na iziphumo ebezingalindelekanga, kubalulekile ukuba uqhagamshelane nomboneleli wakho wezempilo.
(2) Izilumkiso xa uthatha i-Tadalafil Powder:
Gwema ukudibanisa i-Tadalafil Powder kunye neziyobisi ze-antihypertensive, i-cannabis, ubuninzi botywala, ukutya okunamafutha, kunye neemveliso eziqulethe ijusi ye-grapefruit.
Yintoni enye ebalulekileyo ukuba uyazi malunga nokuthatha i-Tadalafil Powder?
ubudala
I-Cialis inokuhlala ixesha elide kwabanye abantu abangaphezu kweminyaka engama-65 ngenxa yokuba umzimba wakho uthatha ixesha elide ukucubungula iyeza. Oku kuchaphazela indlela ephuma ngokukhawuleza ngayo emzimbeni wakho.
Amanqanaba eCialis emzimbeni wakho anokuphakama ngenxa yokusebenza kakubi kwezintso, ukuphakamisa imiphumo emibi. Kule meko, ugqirha wakho unokulungelelanisa umthamo wakho.
Isifo senhliziyo kunye nezinye iimeko
Ukuba uneminyaka engaphezu kwe-65, unesifo senhliziyo, okanye unengxaki yesibindi okanye izintso, ugqirha wakho unokufuna ukulungelelanisa umthamo wakho we-Cialis kwaye ujonge indlela amayeza asebenza ngayo kuwe.
I-Cialis yobuxoki
Thenga iipilisi zeCialis kuphela ngomyalelo kagqirha. Amayeza e-PDE5 aphakathi kwawona mayeza omgunyathi axhaphakileyo asasazwa kwi-Intanethi. Zinokuyibeka emngciphekweni impilo-ntle yomntu. Ukuba ufuna ukuthenga i-Tadalafil Powder bulk ukuvelisa iipilisi, hlala ukhumbula ukuthenga i-Tadalafil Powder kumthengisi othembekileyo. Umthengisi othembekileyo onjenge-AASRAW uya kubonelela ngeengxelo ezivavanyiweyo ezifana ne-COA, i-HPLC kunye ne-NMR
Thatha kanye njengoko kuyalelwe.
I-Cialis kufuneka ithathwe ngokuchanekileyo njengoko ilawulwa ngugqirha wakho. Ukuthintela iziphumo ebezingalindelekanga, musa ukuthatha iidosi ezongezelelweyo okanye utshintshe ishedyuli yakho yedosi ngaphandle kokubonisana nogqirha wakho kuqala.
Kuphi ukuthenga iTadalafil Powder kwi-wholesale?
Umthombo oThembekileyo we-FDA ulumkisa ukuba ezinye iikhemesti ezikwi-Intanethi azingababoneleli abathembekileyo. Umntu kufuneka ahlale ejonga uphononongo lweTadalafil kwaye aqaphele iimpawu zekhemesti ethembekileyo. Ukufumana phi ukuphononongwa kwePowder ye-Tadalafil eyinyani kunye nethembekileyo kunye nomthombo? Mhlawumbi ungazama ukujonga ngeReddit. I-Cialis ifumaneka kuphela ngomyalelo. Nangona kunjalo, yethu i-Tadalafil Powder iyisithako esisebenzayo se-Cialis, unokufumana ezininzi i-Tadalafil Powder umthengisi kwi-intanethi. Kukho ezininzi i-Tadalafil Powder ezithengiswa kwi-intanethi, kubalulekile ukufumana umthengisi wangempela kunye nothembekileyo. I-AASRAW ngumenzi omnye othengisa umgangatho ophezulu weTadalafil Powder. I-Tadalafil Powder i-wholesale trades ixhaphake kakhulu kuneentengiso zokuthengisa njengoko ngokuqhelekileyo kuthengwa ngobuninzi ngokuthe ngqo kwi-factory. Thenga i-Tadalafil Powder Wholesale kwi-AASRAW iya kufumana ixabiso elihle.
Ingxelo yoVavanyo lwePowder yeTadalafil-HNMR
Yintoni i-HNMR kwaye Ikuxelela ntoni i-spectrum ye-HNMR?H I-Nuclear Magnetic Resonance (NMR) ispectroscopy bubuchule bokuhlalutya bekhemistri esetyenziswa kulawulo lomgangatho kunye nophando lokumisela umxholo kunye nokusulungeka kwesampulu kunye nobume bayo bemolekyuli. Umzekelo, i-NMR inokuhlalutya ngokobungakanani imixube equlathe iikhompawundi ezaziwayo. Kwiikhompawundi ezingaziwayo, i-NMR inokusetyenziselwa ukuthelekisa ngokuchasene neelayibrari ezibonwayo okanye ukuqikelela ulwakhiwo olusisiseko ngokuthe ngqo. Nje ukuba ulwakhiwo olusisiseko lwaziwe, i-NMR inokusetyenziselwa ukumisela ulungelelwaniso lwemolekyuli kwisisombululo kunye nokufunda iipropathi ezibonakalayo kwinqanaba lemolekyuli ezifana notshintshiselwano oluhambelanayo, utshintsho lwesigaba, ukunyibilika, kunye nokusasazwa.
I-Tadalafil powder (171596-29-5)-COA
I-Tadalafil powder (171596-29-5)-COA
Indlela yokuthenga Tadalafil Umgubo ovela kwi-AASraw?
❶Ukuqhagamshelana nathi ngenkqubo yethu yokubuza nge-imeyile, okanye usishiyele inombolo yakho ka-whatsapp, ummeli wethu wenkonzo yabathengi (CSR) uya kuqhagamshelana nawe kwiiyure ezili-12.
❷Ukusinika ubungakanani obubuziweyo kunye nedilesi.
❸I-CSR yethu iya kukubonelela ngekoteyishini, ixesha lokuhlawula, inombolo yokulandelela, iindlela zokuthunyelwa kunye nomhla wokufika oqikelelweyo (ETA).
❹Intlawulo yenziwe kwaye iimpahla ziya kuthunyelwa kwiiyure ezili-12.
❺Impahla efunyenweyo kwaye unike izimvo.
Umbhali weli nqaku:
UGqr Monique UHong uthweswe isidanga kwiKholeji yase-UK Imperial yaseLondon kwiFakhalthi yezoNyango
Umbhali wephepha leJenali yeNzululwazi:
1. Emanuel Fryk
ISebe leMolekyuli kunye neClinical Medicine, iZiko lezoNyango, iSahlgrenska Academy, iYunivesithi yaseGothenburg, eSU Sahlgrenska, 413 45 Gothenburg, Sweden
2. Dorota Rogacka
ISebe le-Molecular Biotechnology, iFaculty of Chemistry, iYunivesithi yaseGdansk, iWita Stwosza 63, Gdansk 80-308, Poland
3. E. Deconinck
Ulwalathiso lwezeNzululwazi kwiMingcipheko yeMichiza kunye neMpilo yeMpilo, iNkonzo yaMayeza kunye neeMveliso zezeMpilo, iSciensano, J. Wytsmanstraat 14, B-1050, Brussels, Belgium
4. Iman Shamohammadi
ISebe le-Urology, iSibhedlele saseNemazee, iYunivesithi yaseShiraz yeSayensi yezoNyango, eShiraz, e-Iran
5. Natsumi Tomita
Isebe leSibhedlele seKhemesti, iSikole seSifundo seSayensi, iYunivesithi yaseNagoya City, 3-1 Tanabe do-ri, Mizuho-ku, Nagoya 467-8603, Japan
Abagqirha okanye izazinzulu azikukhuthazi nangayiphi na indlela ukuthengwa, ukuthengiswa, okanye ukusetyenziswa kwale mveliso nangasiphi na isizathu. I-Aasraw ayinayo indibaniselwano okanye ubudlelwane, ichazwa okanye ngenye indlela, ngala magqirha. Injongo yokucaphula kukuvuma kunye nokuncoma uphando olupheleleyo kunye nomsebenzi wophuhliso owenziwe ngoososayensi abasebenza kule nto.
isingqiniso
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[2] Sebastianelli A, Spatafora P, Morselli S, Vignozzi L, Serni S, McVary KT, Kaplan S, Gravas S, Chapple C, Gacci M. "I-Tadalafil Yedwa okanye ngokudibanisa neTamsulosin yoLawulo lwe-LUTS / BPH kunye ne-ED . "Curr Urol Rep. 2020 Okt 27;21(12):56. doi: 10.1007/s11934-020-01009-7. PMID: 33108544
[3] Ruopp NF, Cockrill BA. "Ukuxilongwa kunye noNyango lwe-Pulmonary Arterial Hypertension: Uphononongo." JAMA. 2022 Epreli 12; 327 (14): 1379-1391. doi: 10.1001/jama.2022.4402. PMID: 35412560
[4] Sitbon O, Cottin V, Canuet M, Clerson P, Gressin V, Perchenet L, Bertoletti L, Bouvaist H, Picard F, Prévot G, Bergot E, Simonneau G. “Unyango oludityanisiweyo lokuqala lwe-macitentan kunye ne-tadalafil kwi-pulmonary arterial uxinzelelo lwegazi."Eur Respir J. 2020 Sep 3;56(3):2000673. doi: 10.1183/13993003.00673-2020. Shicilela ngo-2020 Septemba PMID: 32350101
[5] Prasetyo DT, Raharja PAR, Mantiri BJ, Ringoringo DRL, Rahman IA, Felizio J, Tambunan MP, Fadhly SF, Rahardjo HE. "I-Tadalafil Kanye ngoSuku lwaMadoda ane-Erectile Dysfunction: Ngaba iPhakamileyo kunoLawulo lwe-On-Demand?" I-Acta Med Indones. 2019 Jul; 51(3): 275-281. PMID: 31699953
[6] Banjac NM, Vasović VM, Stilinović NP, Prodanović DV, Tomas Petrović AD, Vasović LV, Jakovljević VL. "I-Tadalafil kwi-Doses eNyusayo: Impembelelo kwi-Coronary Blood Flow kunye ne-Oxidative Stress kwi-Isolated Rat Hearts." I-Pharmacology. 2022;107(3-4):150-159. doi: 10.1159/000520498. Epub 2021 Dec 10. PMID: 34903698