Ingcaciso yeMveliso
Isiqulatho
1.Vardenafil Hydrochloride Powder ividiyo-AASraw
I-2.Raw Vardenafil HCL Powder Basic Characters
3.Ingxelo yokuHlola i-Vardenafil ye-HCL yePowder eluhlaza-HNMR
4.Yintoni iVardenafil Hydrochloride (Vardenafil HCL) Powder?
5.Isebenza njani iVardenafil HCL?
6.Ngaba iVardenafil HCL iyasebenza kuzo zonke iintlobo ze-erectile dysfunction?
7.I-Vardenafil HCL ihlala ixesha elingakanani?
I-8.I-Vardenafil HCL Powder ithelekisa njani ne-powder efanayo ye-enchaner yesini?
9.Ziziphi iimpembelelo zeVardenafil HCL?
10.Summary
11.Iinkcazo
I-12.Indlela yokuthenga i-Vardenafil HCL Powder esuka kwi-AASraw?
1. IVardenafil Hydrochloride Ividiyo yomgubo-AASraw
2. ekrwada Vardenafil HCL Iimpawu zePowder Basic
igama: | UVardenafil hydrochloride (Levitra) powder |
CAS: | 224785-91-5 |
Ifomula yeMolekyuli: | C22H19N3O4 |
Ubunzima Ezinto: | 389.4 |
Melt Point: | 298-300 ° C |
Isitoreji sokugcina: | 20ºC |
umbala: | Powder |
3. ekrwada Vardenafil HCL Ingxelo yoVavanyo lwePowder-HNMR
Yintoni i-HNMR kwaye ikuxelela ntoni i-spectrum ye-HNMR? H I-Nuclear Magnetic Resonance (NMR) ispectroscopy bubuchule bohlalutyo lwekhemistri esetyenziswa kulawulo lomgangatho kunye nophando lokufumanisa umxholo kunye nokusulungeka kwesampulu kunye nokwakheka kwemolekyuli. Umzekelo, i-NMR inokuhlalutya ngokobungakanani imixube equlathe iikhompawundi ezaziwayo. Kwiikhompawundi ezingaziwayo, i-NMR inokusetyenziselwa ukuthelekisa ngokuchasene neelayibrari ezibonwayo okanye ukuqikelela ulwakhiwo olusisiseko ngokuthe ngqo. Nje ukuba ulwakhiwo olusisiseko lwaziwe, i-NMR inokusetyenziselwa ukumisela ulungelelwaniso lwemolekyuli kwisisombululo kunye nokufunda iipropathi ezibonakalayo kwinqanaba lemolekyuli ezifana notshintshiselwano oluhambelanayo, utshintsho lwesigaba, ukunyibilika, kunye nokusasazwa.
4.Yintoni iVardenafil Hydrochloride (Vardenafil HCL) Powder?
I-Vardenafil Hydrochloride ingeyeklasi yeziyobisi ezibizwa ngokuba yi-phosphodiesterase type 5 inhibitors, eyaziwa ngokuba yi-PDE-5 inhibitors. Kule nqaku, siya kubhekisela kuVardenafil HCL njengegama elifutshane.
UVardenafil uyaziwa nangokuthi nguLevitra okanye uStaxyn. Nokuba yeyiphi na igama lebhrendi, eli yeza lisebenza injongo enye: ukunceda amadoda ukuba anqobe ukungasebenzi kakuhle kwe-erectile kube kanye.
I-AASraw inikezela nge-vardenafil yangempela ye-HCL i-powder bulk ye-erectile dysfunction kwaye iye yaziwa ngabaninzi ababoneleli abathengisa iipilisi ze-vardenafil hcl okanye ii-capsules, banike iimpendulo ezintle kwi-Vardenafil HCL powder ecocekileyo.
5.Isebenza njani iVardenafil HCL?
I-Vardenafil HCL kunye nezinye i-PDE5 inhibitors zisebenza ngokunyusa ukuhamba kwegazi kwi-penis ukuphatha i-ED. Ukuqonda indlela asebenza ngayo la machiza kuncediswa kukuqonda inkqubo yokwakhiwa.
Xa uvuselelwa ngokwesondo, ingqondo yakho ithumela umqondiso kwimithambo yegazi kwilungu lobudoda bakho, ibangele ukuba ikhuphe ikhemikhali ebizwa ngokuba yinitric oxide. I-nitric oxide isasazeka kuyo yonke imithambo yegazi, ivuselela ukwakheka kwenye imolekyuli eyaziwa ngokuba yi-cGMP. I-cGMP iphumza imithambo yegazi kwilungu lakho lobudoda, ivumela igazi elingakumbi ukuba lingene kwizicubu zayo.
I-Vardenafil HCL inqanda i-PDE5 enzyme, ejongene nokuqhekeka kwe-cGMP. Ukuthintela le enzyme iphakamisa inqanaba le-cGMP kwimithambo yegazi yakho, ivumela igazi elininzi ukuba limpompoze kwilungu lakho lobudoda.
6.Ngaba iVardenafil HCL iyasebenza kuzo zonke iintlobo ze-erectile dysfunction?
I-ED yimeko entsonkothileyo enezizathu ezahlukahlukeneyo, kuquka ukungalingani kwehomoni okubangelwa kukungahambi kakuhle kwegazi, uxinzelelo, ukuxhalaba, ukudakumba, kunye nokungasebenzi kakuhle kwemithambo-luvo.
I-Vardenafil kunye nezinye i-PDE5 inhibitors zisetyenziswa rhoqo njengonyango lokuqala xa kukrokrelwa izizathu zomzimba ze-ED. Kunokuba luncedo, umzekelo, ukuba ukujikeleza kakubi kuhambelana nesifo sikashukela okanye isifo senhliziyo. I-ED yakho yenziwe ngumthombo othembekileyo. I-PDE5 inhibitors ayisebenzi ekuphatheni i-ED ebangelwa yimiba yengqondo efana noxinzelelo okanye ukuxhalaba. Ukuba izizathu zengqondo zikrokrelwa, ugqirha unokuncoma unyango lwengqondo.
7.I-Vardenafil HCL ihlala ixesha elingakanani?
I-Vardenafil HCL, unyango lwe-ED, inokuthatha naphi na ukusuka kwi-25 ukuya kwi-60 imizuzu ukuya emsebenzini. Gcina ukhumbula, nangona kunjalo, ukuba uya kuba nakho ukufumana i-erection kuphela ukuba kukho ukuvuselela ngokwesondo. Awuyi kuba nokwakhiwa nasemva kwemizuzu engama-60 ukuba akukho vuselelo lwesondo. Iyeza liya kusebenza emzimbeni wakho iiyure ezisibhozo ukuya kwezilishumi.
I-8.I-Vardenafil HCL Powder ithelekisa njani ne-powder efanayo ye-enchaner yesini?
I-Vardenafil HCL powder yi-PDE5 inhibitor, efana ne-sildenafil citrate (Viagra). Yesibini echazwe ngokuqhelekileyo iyeza le-erectile dysfunction (kwindawo yesibini kwi-Viagra). I-Vardenafil HCL powder isebenza ngokufanayo ne-sildenafil citrate ekubeni ikhulula imithwalo yegazi kwi-penis, ivumela ukunyuka kwegazi kunye nokwakhiwa.
Kukho iiyantlukwano ezimbalwa phakathi kwala mayeza mabini, nangona kunjalo, okwenza i-Vardenafil HCL powder ibe nomtsalane ngakumbi:
♦ I-Vardenafil HCL powder ingathathwa njengoko ifunekayo; akuyimfuneko ukuyithatha yonke imihla okanye ngeveki.
♦ Ugqirha wakho unokumisela i-Vardenafil HCL kwi-dose ephantsi kunokuba wayeya kuba sildenafil citrate.
9.Ziziphi iimpembelelo zeVardenafil HCL?
Ukunciphisa umngcipheko wemiphumo emibi, nceda wazise umboneleli wakho wezonyango malunga nawo onke amayeza owathathayo, kubandakanywa neyeza kunye neyeza-counter-the-counter, iivithamini, kunye nezongezelelo zemifuno.
Ngaphezulu kweminyaka eyi-20 kwiimarike, kukho ulwazi oluninzi malunga nemiphumo emihle ye-Vardenafil HCL kwi-erectile dysfunction kunye nemiphumo yayo.
Ezi zilandelayo ziziphumo zecala eziqhelekileyo zeVardenafil HCL:
▪ Intloko ebuhlungu
▪ Ukugungxulwa kolusu
▪ isisu esibuhlungu
▪ Umbono ongaqhelekanga okanye oluzizi
▪ Impumlo ebalekayo okanye exineneyo
▪ Umqolo okanye izihlunu ezibuhlungu
▪ Ukuba nesiyezi nesicaphucaphu
▪ Irhashalala
Ezinye iziphumo ebezingalindelekanga zinokwenzeka. Ukuba nayiphi na kwezi okanye ezinye iziphumo ebezingalindelekanga ziyakukhathaza okanye ungahambi, yeka ukuthatha iyeza, qhagamshelana nomboneleli wakho wezempilo, okanye ufune unyango olungxamisekileyo.
10.Summary
I-Vardenafil Hydrochloride iyingxenye ye-PDE-5 inhibitors kwaye sihlala siyisebenzisa ukuphatha ingxaki ye-ED eyabangelwa yimiba yenyama efana nokujikeleza kakubi.
I-AASraw ngumvelisi oqeqeshiweyo we-Vardenafil HCL powder ene-lab ezimeleyo kunye nefektri enkulu njengenkxaso, yonke imveliso iya kwenziwa phantsi kolawulo lweCGMP kunye nenkqubo yokulawula umgangatho olandelwayo. Inkqubo yokubonelela izinzile, zombini ii-odolo zokuthengisa kunye nee-wholesale zamkelekile.
11.Ingxelo
[1] Bódi B, et al. Ixesha elide i-PDE-5A inhibition iphucula umsebenzi we-Myofilament kwi-Cardiomyocytes ye-Ventricular yasekhohlo kunye ne-Right ngokusebenzisa iindlela ezahlukeneyo ezihlukeneyo kwiiNtliziyo ze-Diabetic Rat. Antioxidants (Basel). 2021 Nov 6. 10 (11): 1776. [2] Wayman C, Phillips S, Lunny C, Webb T, Fawcett L, Baxendale R et al. I-Phosphodiesterase 11 (PDE11) ukulawulwa kwe-spermatozoa physiology. Int J Impot Res 2005; 17: 216–223 . [3] Shabsigh R, Burnett AL, Eardley I, Sharlip ID, Ellsworth PI, Garcia CS et al. Ixesha ukusuka kwi-dosing ukuya kwimizamo yokulala ngesondo kumadoda athatha i-tadalafil kwizilingo zeklinikhi. BJU Int 2005; 96: 857–863. [4] Oudot A, et al. Ukudibanisa kwe-BAY 60-4552 kunye ne-vardenafil yenza i-proerectile facilitator imiphumo kwiigundane ezinokulimala kwe-nerve cavernous: ubungqina bokufunda ingcamango yonyango lwe-phosphodiesterase uhlobo lwe-5 inhibitor failure. I-Eur Urol. 2011 Nov. 60(5):1020-6. [5] Gresser U, et al. Ukungasebenzi kakuhle kwe-Erectile: ukuthelekiswa kokusebenza kunye nemiphumo emibi ye-PDE-5 inhibitors sildenafil, i-vardenafil kunye ne-tadalafil-uphononongo loncwadi. I-Eur J Med Res. 2002 Oktobha 29. 7(10): 435-4612. Indlela yokuthenga i-Vardenafil HCL Powder kwi-AASraw?
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